Anastrozole – Arimidex
Aromatase Inhibitor tablets designed for the reduction and elimination of estrogen levels.
Anastrozole, commonly known as Arimidex, is a potent aromatase inhibitor (AI) that falls into the anti-estrogen category. Unlike Nolvadex and Clomid, which are selective estrogen receptor modulators (SERMs), aromatase inhibitors address estrogen metabolism through a distinct mechanism.
Why Use Anastrozole
Anastrozole is the leading AI favored in the bodybuilding community due to its effectiveness in managing various estrogen-related side effects, such as:
- bloating
- gynecomastia
- water retention
- high blood pressure
Best Use
While Nolvadex and Clomid serve as anti-estrogens by occupying receptor sites to block estrogen activity, they do not reduce total estrogen levels. In contrast, aromatase inhibitors like Anastrozole work by binding to the aromatase enzyme to halt the conversion of testosterone into estrogen, effectively lowering estrogen levels in the body.
Anastrozole Cycles
Using Anastrozole daily at 0.5mg (half a tablet) can decrease circulating estrogen levels by up to 50%. For those on cycle, a regimen of 0.5mg every other day can help mitigate estrogen side effects effectively throughout the cycle.

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