Oxymetholone – Anadrol
Anadrol (oxymetholone) is a powerful synthetic steroid available in tablet form. This potent oral anabolic and androgenic compound significantly enhances nitrogen balance, particularly when caloric intake meets adequate levels. Its effects mirror those of testosterone, yet it may lead to severe sexual and physical growth impairments in children, often causing grotesque physical features and sexual dysfunction.
Pharmacology
Anadrol, marketed as Oxymetholone, has an approximate half-life of 8-10 hours, allowing it to remain in the body 2-4 times longer due to its affinity for fatty tissues. Detectable in the system for up to 2 months post-administration, many bodybuilders avoid this compound, opting to use it as an off-season strategy for muscle building.
Indications
In medical settings, Anadrol is prescribed for various types of anemias, including iron deficiency anemia, acquired aplastic anemia, congenital aplastic anemia, myelofibrosis, and anemia related to immunosuppressive treatments. It should be noted that Anadrol is not a substitute for iron, blood transfusions, vitamins, folic acid, or other essential nutrients and is only employed when other supportive treatments are ineffective.
Furthermore, Anadrol is sometimes used to combat HIV-related wasting and severe osteoporosis; however, due to potential side effects, its prescription is becoming less common.
Dosage
The prescribed dose of Anadrol is contingent on body weight, typically ranging from 1.5-2mg/kg (50-200mg/week) for both adults and children. Responses to treatment may take 2-3 weeks or more, with some patients requiring lower doses for ongoing efficacy in treating aplastic anemias. Anadrol is exclusively available in tablet form and is not administered intravenously.
Side Effects
Before commencing Anadrol, be aware of its extensive side effects:
- Jaundice
- Potential for liver cancer
- Penile enlargement if taken prepuberty
- Testicular atrophy and reduced sperm count post-puberty
- Impotence and painful erections
- Clitoral enlargement and menstrual irregularities in women
- Insomnia
- Gynecomastia
- Voice deepening
- Increased hair growth
- Fatigue
- Body swelling
- Elevated blood sugar levels
Contraindications
- Prostate cancer
- Male breast cancer
- Female breast cancer
- Pregnancy
- Liver issues
- Allergic reactions to the drug
Bodybuilding
Anadrol is popular among athletes and bodybuilders due to its powerful anabolic effects and relative affordability. Easily accessible, it is commonly procured through online sources or forged prescriptions, and often smuggled from countries like Mexico and Thailand.
Orally ingested Anadrol promotes gradual weight gain, with initial effects typically observed after 3-4 weeks, contradicting online claims of rapid results. Maintaining weight gains usually necessitates a minimum duration of 3-6 weeks. Athletes often cycle Anadrol with growth hormone and thyroxin, although water retention is a notable side effect. Nevertheless, many claim this aids joint protection during training.
Furthermore, Anadrol is regarded for its potential to enhance recovery post-injury.
Given its substantial side effects and possible liver cancer risk, its use should be cautious. Bodybuilders commonly alternate Anadrol with other anabolic steroids.
Recent studies indicate that Anadrol can unpredictably affect mental health, with reports of increased anger, irritability, and aggression following extended use.
Bodybuilding dosages are subjective, but most experts recommend starting with 50 mg daily for 2-3 weeks, increasing to 75 mg if results are insufficient. However, it is advisable not to exceed 6-8 weeks of use. Anadrol is available under various brand names, such as Thai 50 or Strol V, but caution is warranted due to concerns over counterfeit products.
Cost
The cost of Anadrol ranges from $150 to $200 for a supply of 100 tablets.
Control
Increasing abuse of Anadrol has led to tighter regulation in North America, where it is classified as a Schedule III controlled substance requiring a valid physician’s prescription. Possession with intent to sell carries significant legal repercussions, including hefty fines and potential imprisonment.
Detection
Strictly prohibited in competitive sports, Anadrol is routinely tested in athletes. A positive result typically signifies suspension. This drug and its metabolites can be detected in urine for 20-45 days after the last dosage.
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