Anastrozole – Arimidex
Aromatase Inhibitor tablets designed for the effective breakdown and reduction of estrogen.
Anastrozole, popularly known as Arimidex, is a powerful aromatase inhibitor (AI) that falls under the anti-estrogen category. Unlike SERMs such as Nolvadex and Clomid, which are Selective Estrogen Receptor Modulators, AIs operate on estrogen metabolism through unique mechanisms.
Reasons to Choose Anastrozole
Anastrozole is highly regarded as it was the pioneering AI in the bodybuilding community. Its primary function is to mitigate virtually all potential estrogen-related side effects, including:
- bloating
- gynecomastia
- water retention
- high blood pressure
Optimal Usage
While Nolvadex and Clomid serve as anti-estrogens by blocking receptor sites to prevent new estrogen formation, AIs like Anastrozole actively reduce existing estrogen levels. The aromatase enzyme, responsible for estrogen conversion, is effectively inhibited by these compounds, leading to a significant decrease in estrogen.
Anastrozole Cycling
Using Anastrozole daily at a dosage of 0.5mg (half a tablet) can decrease circulating estrogen levels by as much as 50%. Therefore, administering 0.5mg every other day during a cycle can help eliminate estrogen-related side effects entirely.
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