Exemestane (Aromasin)
Exemestane, commonly marketed as Aromasin, is a significant pharmaceutical agent primarily used as a treatment for breast cancer. However, it has gained popularity among steroid users to combat estrogenic side effects associated with aromatizable steroids.
As an aromatase inhibitor, Exemestane is classified as an anti-estrogen, similar to others like Anastrozole (Arimidex). In contrast, Selective Estrogen Receptor Modulators (SERMs) like Nolvadex (Tamoxifen) work differently. Both SERMs and AIs effectively address estrogen-related issues, but they have distinct mechanisms of action.
Exemestane functions by inhibiting aromatase, the enzyme responsible for estrogen production. This suppression is crucial for managing breast cancer growth and alleviating the adverse effects stemming from certain steroids used for enhanced performance and physique.
Approved by the FDA in 1999, Exemestane quickly rose to prominence due to its effectiveness in lowering estrogen levels.
Half-Life
Exemestane has a half-life ranging between 24 to 27 hours, indicating that it takes this amount of time for half the active substance to be eliminated from the body. Typically, it can be expected to be cleared within 48 to 54 hours. However, detection times can extend up to 2 weeks in anti-doping tests.
What is Exemestane Used For?
Primarily, Exemestane, sold as Aromasin, is utilized to reduce estrogen levels in the body, mitigating various negative effects associated with excess estrogen. This is particularly beneficial for steroid users seeking protection from estrogenic side effects, as well as for women with hormonally sensitive breast cancer.
As a suicidal aromatase inhibitor, Exemestane irreversibly binds to the aromatase enzyme, permanently inhibiting its effects, unlike other AIs like Arimidex. Studies show Aromasin can reduce estrogen levels by approximately 85%, establishing its efficacy compared to non-suicidal AIs.
Steroid users often experience elevated estrogen levels due to substances like Dianabol and Testosterone, which can lead to serious side effects, including gynecomastia and hypertension. Exemestane effectively controls these issues by lowering estrogen levels.
Dosage
Given the half-life of Exemestane, daily administration is recommended to maintain stable blood levels. Some may opt for an every-other-day schedule to avoid excessive estrogen suppression, depending on individual needs. Dosage typically varies between 12.5 mg every other day to 25 mg daily, but users must be cautious not to overdose, as excessive suppression can lead to its own adverse effects.
Side Effects
While Aromasin (Exemestane) is generally well-tolerated, high dosages can result in low estrogen levels, leading to potential complications such as:
- depression
- insomnia
- impotence
- low energy
To minimize risks, it’s essential to use Exemestane judiciously, adhering to lower dosages for optimal estrogenic protection. Side effects occur infrequently in bodybuilders who typically use short-term doses. Common complaints include sweating, insomnia, headaches, and joint pain, which often diminish with reduced dosage.
Ultimately, failure to use any aromatase inhibitor while taking aromatizable steroids significantly increases the likelihood of experiencing side effects, emphasizing the importance of estrogenic protection.
Anonymous (verified owner) –
Massive difference in workout intensity.
Rongo Y. (verified owner) –
Pretty much what I expected. Good product.
Alexandru P. (verified owner) –
Efeitos fortes. Apenas um pouco inconsistente.
Anonymous (verified owner) –
جودة Euro-Pharmacies Exemestanex bag 50 tabs (20 mg/tab) واضحة على الفور. ممتاز!
Jasur G. (verified owner) –
Работает как рекламировалось. Никаких сюрпризов.
Marcin O (verified owner) –
منتج من الدرجة الأولى. Euro-Pharmacies Exemestanex bag 50 tabs (20 mg/tab) ممتاز.
Mónica R. (verified owner) –
Perfectly dosed. Perfect results.
Min O (verified owner) –
منبهر بالتأثيرات لكنني كنت أتوقع المزيد قليلاً.
Ramin L. (verified owner) –
Found my new supplier for life.
Anonymous (verified owner) –
Been using Euro-Pharmacies Exemestanex bag 50 tabs (20 mg/tab) for months now. Consistent results every time.
Piper X. (verified owner) –
A qualidade de Euro-Pharmacies Exemestanex bag 50 tabs (20 mg/tab) é imediatamente evidente. Excelente!
Anonymous (verified owner) –
非常好的产品。几乎完美。
Anonymous (verified owner) –
This Euro-Pharmacies Exemestanex bag 50 tabs (20 mg/tab) is what winners use.
Anonymous (verified owner) –
Good product. Could be a bit stronger.
Beka U (verified owner) –
منتج متين. يقوم بما يجب أن يقوم به.
Virat K (verified owner) –
效果不错。不能抱怨。
Yerzhan L (verified owner) –
Não vale o dinheiro.
Marija G (verified owner) –
تجربة رائعة مع Euro-Pharmacies Exemestanex bag 50 tabs (20 mg/tab). أوصي به بشدة.
Anonymous (verified owner) –
Very good product. Nearly perfect.
Mauro K. (verified owner) –
تأثيرات ملحوظة من الاستخدام الأول. Euro-Pharmacies Exemestanex bag 50 tabs (20 mg/tab) لا يصدق!
Ulugbek L (verified owner) –
Assez efficace. Presque parfait.
Anonymous (verified owner) –
Will be a lifetime customer now.
Anonymous (verified owner) –
Powerful stuff. Use with caution.
Alexandra Y (verified owner) –
Definitiv überdurchschnittlich.
Hee-jun I. (verified owner) –
Habe bessere Ergebnisse mit viel günstigeren Alternativen erzielt.
Yara H. (verified owner) –
Producto de la más alta calidad. Euro-Pharmacies Exemestanex bag 50 tabs (20 mg/tab) es impecable.
Anonymous (verified owner) –
يقوم بعمله لكنه ليس مثيراً للإعجاب.
Anonymous (verified owner) –
Insane results. Will be stocking up next time.
Alexander C (verified owner) –
مثالي! Euro-Pharmacies Exemestanex bag 50 tabs (20 mg/tab) هو بالضبط ما احتجت إليه.
Sofia J. (verified owner) –
The difference is remarkable.
Anonymous (verified owner) –
Unvergleichliche Qualität. Euro-Pharmacies Exemestanex bag 50 tabs (20 mg/tab) ist einfach das Beste.
Hai Y. (verified owner) –
يعمل جيداً لكنه غالي الثمن مقارنة بالآخرين.
Anonymous (verified owner) –
Pretty strong stuff. Just short of perfect.
Akira P. (verified owner) –
Pretty much what I expected. Good product.
Amangeldi I (verified owner) –
منتج رائع، توصيل سريع. Euro-Pharmacies Exemestanex bag 50 tabs (20 mg/tab) رائع.
Keti S (verified owner) –
Assolutamente consigliato! Euro-Pharmacies Exemestanex bag 50 tabs (20 mg/tab) è un prodotto straordinario.
Zulfiya X. (verified owner) –
Quasi buono come il mio solito marchio.
Anonymous (verified owner) –
Producto sólido. Hace lo que debe hacer.
Rana U. (verified owner) –
Risultati sorprendenti fin dal primo utilizzo di Euro-Pharmacies Exemestanex bag 50 tabs (20 mg/tab).
Marlies N. (verified owner) –
Molto buon prodotto. Quasi perfetto.
Ibrahim T. (verified owner) –
Love this stuff! Works like magic.
Tadeusz J. (verified owner) –
Good product. Does what it says.
Zhiwei A. (verified owner) –
效果不错。不能抱怨。
Spyridon F (verified owner) –
Efficacia sorprendente fin dalle prime applicazioni. Euro-Pharmacies Exemestanex bag 50 tabs (20 mg/tab) è fantastico.
Anonymous (verified owner) –
Presque aussi bon que ma marque habituelle.
Parisa D (verified owner) –
كنت أتوقع أكثر قليلاً مقابل السعر، لكنه جيد رغم ذلك.
Alisher E (verified owner) –
Качество Euro-Pharmacies Exemestanex bag 50 tabs (20 mg/tab) сразу заметно. Идеально!
Anonymous (verified owner) –
Euro-Pharmacies Exemestanex bag 50 tabs (20 mg/tab) هو بالضبط ما كنت أبحث عنه. مثالي!
Anonymous (verified owner) –
持续使用后效果非常好。
Anonymous (verified owner) –
The difference is incredible.
Theodor R. (verified owner) –
Decisamente sopravvalutato per quello che si ottiene.
Babatunde Y (verified owner) –
Top-notch effectiveness.
Anonymous (verified owner) –
Qualité supérieure à la moyenne. Euro-Pharmacies Exemestanex bag 50 tabs (20 mg/tab) est exceptionnel.
Anonymous (verified owner) –
Fire.
Anonymous (verified owner) –
Spectacular improvement in performance.
Johanna J (verified owner) –
مبالغ في تقييمه بالتأكيد مقابل ما تحصل عليه.
Alexis T (verified owner) –
منتج جيد لكن الشحن كان بطيئاً قليلاً.
Anonymous (verified owner) –
Nothing happened. Pure snake oil.