Dapoxetine
Dapoxetine is a powerful medication designed specifically for treating premature ejaculation in men, marketed under the well-known brand name Priligy.
Mechanism of Action
- Dapoxetine is classified as a selective serotonin reuptake inhibitor (SSRI).
- It enhances serotonin availability in the brain by inhibiting its reuptake, leading to better control over ejaculation.
- This increase in serotonin levels significantly extends the duration before ejaculation.
Indications
- Dapoxetine is primarily indicated for the treatment of premature ejaculation in men.
- Intended for men aged 18 to 64 years experiencing rapid ejaculation issues.
Onset of Action
- The onset of dapoxetine occurs rapidly, typically within 1 to 2 hours post-administration.
Duration of Action
- The effects of dapoxetine can last between 4 to 24 hours, varying based on the dosage and the individual’s response.
Dosage
- The standard dosage for dapoxetine ranges from 30 mg to 60 mg, taken as needed.
- The initial recommended dose is usually set at 30 mg, with adjustments made by the healthcare provider based on the patient’s response.
Side Effects
- Common side effects include dizziness, headaches, nausea, drowsiness, fatigue, and dry mouth.
- Less frequently, users might experience hot flashes, increased anxiety, behavioral changes, or alterations in sexual function.
Contraindications
- Dapoxetine is contraindicated in patients with severe renal or hepatic dysfunction, serious heart conditions, epilepsy, bipolar disorder, or those taking monoamine oxidase inhibitors (MAOIs).
- Moreover, it is crucial to avoid the combination of dapoxetine with alcohol to reduce potential side effects.
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